About 31 results found for searched term "GABA Receptor" (0.205 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M28615 | GABAA receptor agent 1 | GABA Receptor |
| GABAA receptor agent 1 is a high affinity ligand for GABAA receptor, with potent anticonvulsant activity. | ||
| M1952 | Methionine | GABA Receptor |
| D-Methionine; MRX-1024 | ||
| Methionine is an effective chemoprotective agent which can also inhibit the neuronal activity through GABAA receptor activation. | ||
| M2005 | (R)-Baclofen | GABA Receptor |
| STX 209; Arbaclofen | ||
| (R)-baclofen, a gamma-aminobutyric acid derivative and agonist at GABA-B receptors, inhibits nerve conduction in the central nervous system and can be used in studies related to spasticity. | ||
| M2347 | (+)-Bicuculline | GABA Receptor |
| d-Bicuculline | ||
| (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels. | ||
| M4013 | Glabridin | GABA Receptor |
| Glabridin, one of the active phytochemicals in licorice extract, binds to and activates the ligand binding domain of PPARγ, as well as the full length receptor. It is also a GABAA receptor positive modulator promoting fatty acid oxidation and improving learning and memory. | ||
| M4019 | Songorine | GABA Receptor |
| Songorine is a diterpenoid alkaloid isolated from the genus Aconite. Songorine is a GABAA receptor antagonist in rat brain and has anticancer, anti-arrhythmia and anti-inflammatory activities. Songorine has potential to be used in epithelial ovarian cancer (EOC) studies. | ||
| M4073 | Ginsenoside-Rc | GABA Receptor |
| Panaxoside Rc | ||
| Ginsenoside Rc is one of the major ginsenosides. Ginsenoside Rc enhances GABA receptor A (GABAA) -mediated ion channel (IGABA) currents. Ginsenoside Rc also inhibited TNF-α and IL-1β expression. | ||
| M4950 | Topiramate | GluR |
| McN 4853; RWJ 17021 | ||
| Topiramate is an anticonvulsant that antagonizes GluR5 receptors and acts as a positive allosteric modulator of GABA receptor-mediated currents. | ||
| M4959 | Pagoclone | GABA Receptor |
| (+)-RP-59037; IP-456; RP-62955; CI-1043 | ||
| Pagoclone, active (+)-enantiomer of the racemate RP 59037, is a partial GABA(A) receptor agonist that used for treatment of panic and anxiety disorders. | ||
| M5378 | Acamprosate calcium | GABA Receptor |
| Calcium N-acetylhomotaurinate | ||
| Acamprosate calcium (Campral EC) is a GABA receptor agonist and glutamate system modulator. | ||
| M5390 | Afloqualone | GABA Receptor |
| Afloqualone is a agonist of GABA receptor . | ||
| M5575 | Dihydroergotoxine mesylate | GABA Receptor |
| Ergoloid mesylates | ||
| Dihydroergotoxine mesylate is a complex of closely related alkaloid salts; Binds with high affinity to the GABAA receptor Cl- channel, producing an allosteric interaction with the benzodiazepine site. | ||
| M5653 | Flumazenil | GABA Receptor |
| Ro 15-1788 | ||
| Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses. | ||
| M5870 | Pentylenetetrazol | GABA Receptor |
| Pentylenetetrazole, Metrazole, pentetrazol | ||
| Pentylenetetrazol displays activity as a central nervous system and respiratory stimulant. It is considered a non-competitive GABA(A) receptor antagonist. | ||
| M6385 | AA 29504 | Others |
| AA 29504 is a positive allosteric modulator of GABA A receptors. | ||
| M6583 | CGP 36216 hydrochloride | Others |
| CGP 36216 hydrochloride is a gABA B antagonist; displays activity at presynaptic receptors. | ||
| M6720 | Etifoxine hydrochloride | GABA Receptor |
| HOE 36-801 | ||
| Etifoxine hydrochloride is a ligand of the translocator protein (TSPO); also GABA A receptor potentiator. | ||
| M6735 | Flupirtine maleate | Potassium Channel |
| Flupirtine maleate is a selective potassium channel opener, NMDA receptor antagonist and GABAA receptor modulator. | ||
| M6744 | Ganaxolone | GABA Receptor |
| CCD 1042 | ||
| Ganaxolone (CCD 1042) is A neuroactive steroid allopregnenolone analogue synthesized orally and is A selective, high-affinity positive sex modulator of γ -aminobutyrate-A (GABAA) receptor with anticonvulsant properties. Gannadone works through different binding sites with benzodiazepine binding sites and can be used in epilepsy studies related to cyclin-dependent kinase-like 5 (CDKL5) deficiency (CDD). | ||
| M6828 | Indiplon | Others |
| Indiplon is a subtype-selective GABA A receptor positive allosteric modulator. | ||
| M6915 | Loreclezole hydrochloride | Others |
| Loreclezole hydrochloride is a subtype-selective GABA A receptor modulator. | ||
| M6961 | MK 0343 | Others |
| MK 0343 is a subtype-selective GABA A receptor partial agonist. | ||
| M7087 | Org 20599 | Others |
| Org 20599 is a positive allosteric modulator and direct agonist of GABA A receptors. | ||
| M7158 | Pregnanolone | Others |
| Pregnanolone is a gABA A receptor positive allosteric modulator. | ||
| M7252 | SB 205384 | GABA Receptor |
| SB 205384 is a gABA A receptor modulator; slows current decay. | ||
| M7381 | TCS 1105 | Others |
| TCS 1105 is a gABA A α2 benzodiazepine receptor agonist. | ||
| M7382 | TCS 1205 | Others |
| TCS 1205 is a subtype-selective GABA A receptor agonist. | ||
| M7420 | TP 003 | Others |
| TP 003 is a functionally selective GABA A receptor (α3 subtype) partial agonist. | ||
| M7441 | U 90042 | Others |
| U 90042 is a gABA A receptor ligand. | ||
| M7442 | U 93631 | GABA Receptor |
| U 93631 is a gABA A receptor antagonist. | ||
| M7691 | Chlormethiazole hydrochloride | GABA Receptor |
| Chlormethiazole hydrochloride is a GABAA agonist; glycine receptor modulator. | ||
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